SCHEMBL3657964

SCHEMBL3657964

COc1ccc(C2(C(C(=O)Nc3ccc(C(=O)O)cc3F)C3CCCCC3)Nc3cc(F)c(F)cc3N2)c(OC)n1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 18/20 0.44
CYP2C9 P11712 7/20 0.43
CYP3A4 P08684 6/20 0.43
CYP2D6 P10635 5/20 0.43
KCNH2 Q12809 2/20 0.40
CYP26A1 O43174 1/20 0.40
RARB P10826 1/20 0.40
RARG P13631 1/20 0.40
PTGFR P43088 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3655181 0.94 NR1H4 (0.47) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3657230 0.85 NR1H4 (0.41) NR1H4
SCHEMBL1841564 0.81 NR1H4 (0.40) NR1H4
SCHEMBL3801443 0.81 NR1H4 (0.56) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL1841219 0.81 NR1H4 (0.38) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3654638 0.81 NR1H4 (0.46) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL1841709 0.79 NR1H4 (0.38) NR1H4CYP2C9CYP3A4CYP2D6CYP26A1
SCHEMBL1839973 0.79 NR1H4 (0.38) NR1H4CYP2C9CYP3A4CYP2D6
SCHEMBL1836831 0.79 NR1H4 (0.36) NR1H4
SCHEMBL1838285 0.79 NR1H4 (0.37) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225221-A2 CARBOXYL- OR HYDROXYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-09-08 EP disclosed
WO-2009080555-A2 CARBOXYL- OR HYDROXYL- SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO disclosed