SCHEMBL3657230

SCHEMBL3657230

COc1ccc(C2(C(C(=O)O)C3CCCCC3)Nc3cc(F)c(F)cc3N2)c(OC)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.41
POLB P06746 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA2 P47869 1/20 0.33
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
MAPK1 P28482 1/20 0.31
DHODH Q02127 2/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30
NR4A2 P43354 1/20 0.30
PRKAG1 P54619 1/20 0.30
PRKAA1 Q13131 1/20 0.30
PRKAB1 Q9Y478 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3801443 0.87 NR1H4 (0.56) NR1H4GABRG2GABRB3GABRA2HPGD
SCHEMBL1841564 0.87 NR1H4 (0.40) NR1H4RAB9ANPC1MAPK1HPGD
SCHEMBL3654638 0.86 NR1H4 (0.46) NR1H4RAB9ANPC1GABRG2GABRB3
SCHEMBL3657964 0.85 NR1H4 (0.44) NR1H4
SCHEMBL1840133 0.84 NR1H4 (0.36) NR1H4
SCHEMBL1843649 0.84 NR1H4 (0.36) NR1H4MAPK1
SCHEMBL3655181 0.83 NR1H4 (0.47) NR1H4DHODHSMN1; SMN2
SCHEMBL1840558 0.83 L3MBTL1 (0.35) NR1H4
SCHEMBL3657013 0.82 NR1H4 (0.48) NR1H4GABRG2GABRB3GABRA2TSHR
SCHEMBL1836831 0.81 NR1H4 (0.36) NR1H4POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225221-A2 CARBOXYL- OR HYDROXYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-09-08 EP disclosed
WO-2009080555-A2 CARBOXYL- OR HYDROXYL- SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO disclosed