SCHEMBL3658658

SCHEMBL3658658

N=C(S)NCc1c(Cl)cccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
AKR1B1 P15121 1/20 0.41
HTT P42858 3/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2D6 P10635 1/20 0.40
GLA P06280 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
P2RX7 Q99572 3/20 0.39
BACE1 P56817 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PLA2G1B P04054 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL17707535 0.98 HTT (0.42) CYP1A2CYP3A4CYP2C9CYP2C19AKR1B1
SCHEMBL5068038 0.80 NPC1 (0.61) CYP3A4CYP2C9CYP2C19HTTLMNA
SCHEMBL5798047 0.79 AKR1B1 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19AKR1B1
Hydrochloric Acid SCHEMBL4797245 0.79 NPC1 (0.59) CYP3A4CYP2C9CYP2C19HTTLMNA
Hydrochloric Acid SCHEMBL3658158 0.76 ROCK2 (0.38) HTTNPSR1P2RX7BACE1GAA
Bromide SCHEMBL5552280 0.76 ROCK2 (0.38) HTTP2RX7BACE1GAAROCK2
Hydrochloric Acid SCHEMBL11691645 0.74
SCHEMBL2810297 0.74
SCHEMBL5065168 0.73 HTR3E (0.51) LMNAPLA2G1BMAPTATG4BNPC1
SCHEMBL5798053 0.72 AKR1B1 (0.47) CYP1A2CYP3A4CYP2C9CYP2C19AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227457-A2 CHIRAL 3-(BENZYLSULFINYL)-5,5-DIMETHYL-4,5-DIHYDROISOXAZOLE DERIVATIVES AND 5,5-DIMETHYL-3-Ý(1H-PYRAZOL-4-YLMETHYL)SULFINYL¨-4,5-DIHYDROISOXAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND USE OF SAME AS HERBICIDES AND PLANT GROWTH REGULATORS Bayer CropScience AG (DE) 2010-09-15 EP disclosed
WO-2009068171-A2 CHIRAL 3-(BENZYLSULFINYL)-5,5-DIMETHYL-4,5-DIHYDROISOXAZOLE DERIVATIVES AND 5,5-DIMETHYL-3-[(1H-PYRAZOL-4-YLMETHYL)SULFINYL]-4,5-DIHYDROISOXAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND USE OF SAME AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2009-06-04 WO disclosed