SCHEMBL3659618

SCHEMBL3659618

CCOC(=O)c1ccc(NC(=O)C(C2CCCCC2)C2(c3ccc(Cl)cc3)Nc3cc(F)c(F)cc3N2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MAPT P10636 6/20 0.44
RAB9A P51151 4/20 0.43
NPC1 O15118 1/20 0.43
NR1H4 Q96RI1 3/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
POLB P06746 2/20 0.42
HTT P42858 2/20 0.42
ALDH1A1 P00352 1/20 0.42
TRPV1 Q8NER1 2/20 0.41
ABL1 P00519 1/20 0.40
RIN1 Q13671 1/20 0.40
TP53 P04637 1/20 0.40
MEN1 O00255 1/20 0.40
CASP3 P42574 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3661087 0.93 NPSR1 (0.48) GAASMN1; SMN2NPSR1MAPTRAB9A
SCHEMBL3661070 0.90 MAPT (0.47) GAAMAPTRAB9ANPC1TSHR
SCHEMBL3653916 0.88 NR1H4 (0.45) GAASMN1; SMN2NPSR1MAPTNR1H4
SCHEMBL3656516 0.87 NR1H4 (0.46) GAASMN1; SMN2NPSR1MAPTNR1H4
SCHEMBL3652179 0.87 NR1H4 (0.53) SMN1; SMN2MAPTRAB9ANPC1NR1H4
SCHEMBL1843552 0.85 TSHR (0.39) MAPTNR1H4CYP3A4CYP2D6CYP2C9
SCHEMBL1842727 0.85 TSHR (0.39) MAPTNR1H4CYP3A4CYP2D6CYP2C9
SCHEMBL3661109 0.83 MAPT (0.43) NPSR1MAPTRAB9ANPC1TSHR
SCHEMBL3655058 0.82 NR1H4 (0.54) SMN1; SMN2MAPTRAB9ANPC1NR1H4
SCHEMBL1837083 0.82 GAA (0.39) GAASMN1; SMN2NPSR1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225221-A2 CARBOXYL- OR HYDROXYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-09-08 EP disclosed
WO-2009080555-A2 CARBOXYL- OR HYDROXYL- SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO disclosed