SCHEMBL3660185

SCHEMBL3660185

COc1c(Cl)cncc1C#N

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.40
CYP11B1 P15538 5/20 0.40
PRKCQ Q04759 6/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
SRC P12931 3/20 0.37
PDE4D Q08499 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19063459 0.78 PDE4D (0.42) PDE4D
SCHEMBL3825639 0.75 CYP11B2 (0.39) CYP11B2CYP11B1PRKCQ
SCHEMBL15390332 0.74 SRC (0.34) CYP11B2CYP11B1PRKCQSRC
SCHEMBL1920551 0.74 CYP11B2 (0.40) CYP11B2CYP11B1
SCHEMBL27659861 0.72 L3MBTL1 (0.44) L3MBTL1SRC
SCHEMBL1922370 0.72 PRKCQ (0.39) CYP11B2CYP11B1PRKCQSRCPDE4D
SCHEMBL2761020 0.71 CYP11B2 (0.45) CYP11B2CYP11B1
SCHEMBL23291787 0.71 CSNK1A1 (0.40) CYP11B2CYP11B1
SCHEMBL13747989 0.71 CYP11B2 (0.35) CYP11B2CYP11B1
SCHEMBL21718417 0.71 CYP11B2 (0.35) CYP11B2CYP11B1PRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231663-A2 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AS C-MET INHIBITORS Amgen, Inc (US) 2010-09-29 EP disclosed
WO-2009091374-A2 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AMGEN INC. (US) 2009-07-23 WO disclosed