SCHEMBL3660232

SCHEMBL3660232

Cc1c[nH]c(-c2ccc(Nc3ncc4c(n3)C(c3cccc(C(F)(F)F)c3)CCC4)cc2F)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
NLRP3 Q96P20 1/20 0.38
ULK1 O75385 1/20 0.36
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
AXL P30530 1/20 0.35
TYRO3 Q06418 1/20 0.35
MERTK Q12866 1/20 0.35
CTSC P53634 3/20 0.35
PTK2 Q05397 1/20 0.34
PTK2B Q14289 1/20 0.34
CDK2 P24941 3/20 0.34
CDK1 P06493 3/20 0.34
CCNB1 P14635 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3662998 0.93 ULK1 (0.37) ULK1PSEN1PSEN2APH1BNCSTN
SCHEMBL3664169 0.90 PLK1 (0.42) ALDH1A1HPGDRAB9ANLRP3ULK1
SCHEMBL3662338 0.90 PSEN1 (0.44) ULK1PSEN1PSEN2APH1BNCSTN
SCHEMBL1617250 0.82 PSEN1 (0.56) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3663840 0.79 PSEN1 (0.50) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3661349 0.79 PSEN1 (0.40) ULK1PSEN1PSEN2APH1BNCSTN
SCHEMBL3662460 0.78 PSEN1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1617546 0.76 PSEN1 (0.57) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3656955 0.75 CDK2 (0.37) ULK1PTK2CDK2CCNA2PLK1
SCHEMBL3666797 0.75 PSEN1 (0.39) ULK1PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231629-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-09-29 EP disclosed
WO-2009087127-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-07-16 WO disclosed