SCHEMBL3662998

SCHEMBL3662998

Cc1c[nH]c(-c2ccc(Nc3ncc4c(n3)C(c3cc(C(F)(F)F)cc(C(F)(F)F)c3)CCC4)cc2F)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 3/20 0.37
PTK2B Q14289 2/20 0.35
PTK2 Q05397 1/20 0.35
CDK1 P06493 3/20 0.35
CCNT1 O60563 1/20 0.35
CDK4 P11802 1/20 0.35
CCNB1 P14635 1/20 0.35
CCND1 P24385 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
FLT3 P36888 4/20 0.34
KIT P10721 3/20 0.34
CHEK1 O14757 3/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660232 0.93 ALDH1A1 (0.38) ULK1PTK2BPTK2CDK1CCNT1
SCHEMBL3662338 0.89 PSEN1 (0.44) ULK1CDK1CCNB1CDK2PSEN1
SCHEMBL3664169 0.83 PLK1 (0.42) ULK1PTK2PSEN1PSEN2APH1B
SCHEMBL3661349 0.82 PSEN1 (0.40) ULK1CDK1CDK4CCNB1CCND1
SCHEMBL4092721 0.81 PSEN1 (0.54) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3662460 0.79 PSEN1 (0.48) CDK2CDK9PSEN1PSEN2APH1B
SCHEMBL3663840 0.77 PSEN1 (0.50) CDK2PSEN1PSEN2APH1BNCSTN
SCHEMBL3656955 0.77 CDK2 (0.37) ULK1PTK2CDK4CDK2CDK9
SCHEMBL3659216 0.76 PSEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3666797 0.75 PSEN1 (0.39) ULK1PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231629-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-09-29 EP disclosed
WO-2009087127-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-07-16 WO disclosed