SCHEMBL3660244

SCHEMBL3660244

CSc1nc2cc(C(F)(F)F)ccc2s1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
ALOX5 P09917 1/20 0.53
DYRK1A Q13627 2/20 0.52
PPARA Q07869 1/20 0.49
KEAP1 Q14145 1/20 0.47
ILK Q13418 2/20 0.47
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
EPHX2 P34913 1/20 0.44
SCN4A P35499 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PKM P14618 1/20 0.42
NCS1 P62166 1/20 0.42
TOP2A P11388 1/20 0.41
AKR1B1 P15121 1/20 0.40
AGPAT2 O15120 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30602944 1.00 SMN1; SMN2 (0.59) SMN1; SMN2NPSR1ALOX5DYRK1APPARA
SCHEMBL2707227 0.87 PPARA (0.63) SMN1; SMN2NPSR1DYRK1APPARAKEAP1
SCHEMBL17153983 0.87 ALOX5 (0.52) SMN1; SMN2NPSR1ALOX5DYRK1APPARA
SCHEMBL13483968 0.85 SMN1; SMN2 (0.61) SMN1; SMN2NPSR1ALOX5PPARAKEAP1
SCHEMBL17153808 0.82 ALOX5 (0.49) SMN1; SMN2NPSR1ALOX5DYRK1APPARA
SCHEMBL10761623 0.81 DYRK1A (0.60) ALOX5DYRK1APPARAILKCYP1A2
SCHEMBL9393819 0.79 ALOX5 (0.61) SMN1; SMN2ALOX5DYRK1APPARAILK
SCHEMBL1512366 0.78 SMN1; SMN2 (0.65) SMN1; SMN2NPSR1DYRK1APPARAKEAP1
SCHEMBL30602942 0.78 SMN1; SMN2 (0.65) SMN1; SMN2NPSR1DYRK1APPARAKEAP1
SCHEMBL9853857 0.78 POLB (0.56) SMN1; SMN2ALOX5DYRK1AILKEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116926578-A Method for synthesizing heteroaryl thiophenol 新疆大学 2023-10-24 CN disclosed
US-11535607-B2 Isoindolines as HDAC inhibitors VALO HEALTH, INC. (US) 2022-12-27 US disclosed
US-20210253555-A1 ISOINDOLINES AS HDAC INHIBITORS VALO EARLY DISCOVERY, INC. (US) 2021-08-19 US disclosed
US-7897627-B2 Heteroaryl derivatives as orexin receptor antagonists HOFFMANN-LA ROCHE INC. (US) 2011-03-01 US disclosed
US-7897627-B2 Heteroaryl derivatives as orexin receptor antagonists HOFFMANN-LA ROCHE INC. (US) 2011-03-01 US disclosed
US-7897627-B2 Heteroaryl derivatives as orexin receptor antagonists HOFFMANN-LA ROCHE INC. (US) 2011-03-01 US disclosed
EP-2234999-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2010-10-06 EP disclosed
WO-2009080533-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO disclosed
WO-2009080533-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO disclosed
US-20090163485-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-06-25 US disclosed
US-20090163485-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-06-25 US disclosed
US-20090163485-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-06-25 US disclosed
US-5108887-A Zeromethine merocyanine dyes as J-aggregating spectral sensitizers for tabular emulsions E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11535607-B2 Isoindolines as HDAC inhibitors HDAC1, HDAC2, HDAC3 SMN1; SMN2 3655/4885NPSR1 2275/4885ALOX5 4365/4885
US-20090163485-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS HCRTR1, HCRTR2, MTNR1A SMN1; SMN2 2577/4885NPSR1 12/4885ALOX5 272/4885
US-20210253555-A1 ISOINDOLINES AS HDAC INHIBITORS HDAC1, HDAC2, HDAC3 SMN1; SMN2 3655/4885NPSR1 2275/4885ALOX5 4365/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.