SCHEMBL3660786

SCHEMBL3660786

CCCC1(c2ccccc2)NC(=O)N(CC(=O)c2ccc(NC(=O)Cc3ccc(F)cc3)cc2)C1=O

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.57
HDAC6 Q9UBN7 1/20 0.54
LMNA P02545 2/20 0.50
MEN1 O00255 2/20 0.49
FPR2 P25090 1/20 0.48
USP2 O75604 1/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
TSHR P16473 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3662782 0.89 KMT2A (0.56) KMT2AHDAC6LMNAMEN1USP2
SCHEMBL3662888 0.87 KMT2A (0.61) KMT2AHDAC6LMNAMEN1USP2
SCHEMBL3660936 0.86 KMT2A (0.60) KMT2AHDAC6LMNAMEN1USP2
SCHEMBL3659519 0.85 MEN1 (0.56) KMT2ALMNAMEN1GAA
SCHEMBL3663347 0.84 KMT2A (0.58) KMT2AHDAC6LMNAMEN1USP2
SCHEMBL3655230 0.82 KMT2A (0.53) KMT2AHDAC6LMNAMEN1USP2
SCHEMBL3662924 0.81 KMT2A (0.51) KMT2AHDAC6LMNAMEN1FPR2
SCHEMBL4121157 0.81 KMT2A (0.55) KMT2AHDAC6LMNAMEN1USP2
SCHEMBL3658360 0.81 LMNA (0.57) KMT2AHDAC6LMNAMEN1USP2
SCHEMBL3663169 0.80 TSHR (0.59) KMT2ALMNAMEN1FPR2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212314-A1 IMIDAZOLIDINE-2,4-DIONE (HYDANTOIN) DERIVATIVES USEFUL AS NPY Y2 RECEPTOR MODULATORS Novartis AG (CH) 2010-08-04 EP disclosed
WO-2009050200-A1 IMIDAZOLIDINE-2,4-DIONE (HYDANTOIN) DERIVATIVES USEFUL AS NPY Y2 RECEPTOR MODULATORS NOVARTIS AG (CH) 2009-04-23 WO disclosed
US-20090099243-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090099243-A1 ORGANIC COMPOUNDS SLCO4C1, SLCO1B1, SLCO1B3 KMT2A 2020/4885HDAC6 715/4885LMNA 2430/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.