SCHEMBL366085

SCHEMBL366085

CS(=O)(=O)NC(=O)c1ccc(COc2ccc(Cl)c(Cl)c2)c(C#N)c1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 18/20 0.58
SCN5A Q14524 3/20 0.58
HDAC8 Q9BY41 1/20 0.44
MCL1 Q07820 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diethylamine SCHEMBL16239867 0.95 SCN9A (0.53) SCN9ASCN5AHDAC8MCL1
SCHEMBL363727 0.87 SCN9A (0.64) SCN9ASCN5AHDAC8MCL1
SCHEMBL16239703 0.83 SCN9A (0.67) SCN9ASCN5AHDAC8
Diethylamine SCHEMBL16239800 0.82 SCN9A (0.59) SCN9ASCN5AHDAC8
SCHEMBL16319332 0.82 SCN9A (0.61) SCN9ASCN5AMCL1
SCHEMBL16240196 0.80 SCN9A (0.77) SCN9ASCN5AMCL1
SCHEMBL10203178 0.75 SCN9A (0.66) SCN9ASCN5AMCL1
SCHEMBL16240228 0.75 SCN9A (0.78) SCN9ASCN5A
SCHEMBL16239619 0.75 SCN9A (0.78) SCN9ASCN5A
SCHEMBL14890261 0.74 NR4A2 (0.64) SCN9ASCN5AHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 16/4885SCN5A 5/4885HDAC8 925/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.