SCHEMBL3662212

SCHEMBL3662212

CC(C)c1ccc(-c2ccc(C(C)(c3ccc(-c4ccc(N)nn4)cc3)C(C)C)cc2)nn1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 4/20 0.44
TLR9 Q9NR96 2/20 0.36
TLR8 Q9NR97 2/20 0.36
TLR7 Q9NYK1 2/20 0.36
JAK2 O60674 1/20 0.32
HSD11B1 P28845 1/20 0.31
FEN1 P39748 1/20 0.31
CHRNA7 P36544 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2990063 0.86 ALOX5AP (0.52) ALOX5APTLR9TLR8TLR7JAK2
SCHEMBL3001060 0.82 ALOX5AP (0.64) ALOX5APTLR9TLR8TLR7JAK2
SCHEMBL17184739 0.76 KEAP1 (0.40) TLR9TLR8TLR7CHRNA7
SCHEMBL480232 0.76 ALOX5AP (0.65) ALOX5APTLR9TLR8TLR7JAK2
SCHEMBL480207 0.76 ALOX5AP (0.65) ALOX5APTLR9TLR8TLR7JAK2
SCHEMBL933581 0.76 NOS3 (0.40) TLR9TLR8TLR7CHRNA7
SCHEMBL2609362 0.75 MAOB (0.43)
SCHEMBL13262239 0.74 ALOX5AP (0.60) ALOX5APTLR9TLR8TLR7
SCHEMBL480220 0.74 ALOX5AP (0.80) ALOX5APJAK2
SCHEMBL480102 0.74 ALOX5AP (0.80) ALOX5APJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170065-A1 DIPHENYL SUBSTITUTED ALKANES Merck Sharp & Dohme Corp. (US) 2010-04-07 EP claimed
WO-2008156721-A1 DIPHENYL SUBSTITUTED ALKANES MERCK & CO., INC. (US) 2008-12-24 WO claimed