SCHEMBL3662260

SCHEMBL3662260

COC(=O)c1ccnc(N(C)c2ccco2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 3/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
HPGD P15428 2/20 0.35
MAPK1 P28482 3/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
CYP1A2 P05177 2/20 0.35
NPC1 O15118 2/20 0.35
TP53 P04637 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
RECQL P46063 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1790483 0.78 MAPK1 (0.43) KMT2AALDH1A1HPGDMAPK1CYP1A2
SCHEMBL3662262 0.69 KDM4E (0.46) KMT2AALDH1A1HPGDMAPK1SMN1; SMN2
SCHEMBL11903207 0.69 HSD17B10 (0.36) KMT2AALDH1A1HSP90AA1HSP90AB1HPGD
SCHEMBL4384494 0.68 MAPK1 (0.46) KMT2AALDH1A1MAPK1CYP1A2NPC1
SCHEMBL164625 0.68 MAPK1 (0.46) ALDH1A1MAPK1CYP1A2NPC1TP53
SCHEMBL1653862 0.68 HSD17B10 (0.34) KMT2AALDH1A1HSP90AA1HSP90AB1HPGD
SCHEMBL30740821 0.68 JAK3 (0.45) ALDH1A1SMN1; SMN2GAAMAPTPOLB
SCHEMBL13728573 0.67 S1PR4 (0.36) KMT2AALDH1A1CYP1A2NPC1RAB9A
SCHEMBL15500861 0.66 MAPT (0.46) ALDH1A1MAPK1CYP1A2NPC1TP53
SCHEMBL22518516 0.66 MAPK1 (0.44) ALDH1A1MAPK1CYP1A2NPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2237669-A2 CHEMICAL COMPOUNDS Syngenta Limited (GB) 2010-10-13 EP disclosed
WO-2009081112-A2 CHEMICAL COMPOUNDS SYNGENTA LIMITED (GB) 2009-07-02 WO disclosed