SCHEMBL366257

SCHEMBL366257

CON(C)C(=O)c1ccc2c(C(=O)OCCN(C)C)c3ccccc3n2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
TDP1 Q9NUW8 2/20 0.42
RAD52 P43351 2/20 0.40
POLB P06746 2/20 0.40
PHLPP2 Q6ZVD8 1/20 0.40
MAPT P10636 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAOA P21397 1/20 0.35
CNR1 P21554 1/20 0.35
DRD4 P21917 1/20 0.35
ACHE P22303 1/20 0.35
HRH2 P25021 1/20 0.35
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365388 0.90 ALDH1A1 (0.49) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL366312 0.89 ALDH1A1 (0.52) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL364892 0.88 ALDH1A1 (0.47) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL365411 0.87 ALDH1A1 (0.53) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL366302 0.86 ALDH1A1 (0.47) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL366412 0.86 ALDH1A1 (0.49) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL364919 0.86 NR4A2 (0.43) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL365040 0.85 ALDH1A1 (0.48) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL364768 0.84 ALDH1A1 (0.46) ALDH1A1TDP1RAD52POLBPHLPP2
SCHEMBL364813 0.84 ALDH1A1 (0.46) ALDH1A1TDP1RAD52POLBPHLPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed