SCHEMBL3662694

SCHEMBL3662694

CC(Cc1cnc2occc2c1)C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.34
HTR1B P28222 4/20 0.33
FFAR1 O14842 1/20 0.33
NTRK1 P04629 1/20 0.33
MMP9 P14780 2/20 0.33
MMP1 P03956 1/20 0.33
FCER2 P06734 1/20 0.33
MMP3 P08254 1/20 0.33
ELANE P08246 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
CPB2 Q96IY4 1/20 0.32
EPHX1 P07099 1/20 0.31
PIK3CD O00329 1/20 0.31
NR3C2 P08235 1/20 0.31
PLA2G10 O15496 1/20 0.31
PLA2G2A P14555 1/20 0.31
PLA2G5 P39877 1/20 0.31
MMP2 P08253 1/20 0.30
MMP8 P22894 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27425951 0.81 HTR1B (0.39) HTR1BMMP9PIK3CDMMP2MMP8
SCHEMBL1873713 0.76 KDR (0.48) SYK
SCHEMBL3662691 0.73 AURKA (0.41) FFAR1NTRK1ELANEPIK3CDNR3C2
SCHEMBL2846208 0.73 RECQL (0.36) PIK3CD
SCHEMBL10855532 0.73 PARP1 (0.39) PARP1HTR1BPIK3CDCYP1A2MAPT
SCHEMBL2847867 0.70 NR4A2 (0.40) CYP1A2SMN1; SMN2
SCHEMBL13548275 0.70 FGFR1 (0.34) HTR1BPIK3CDMAPTSMN1; SMN2
SCHEMBL10557945 0.70 PSMD14 (0.45) NTRK1PIK3CDSMN1; SMN2
SCHEMBL27532006 0.70 S1PR1 (0.43) FFAR1MMP9PIK3CDMMP2CFD
SCHEMBL6639359 0.70 PIK3CD (0.37) PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152670-A1 BRIDGED SIX-MEMBERED RING COMPOUNDS Actelion Pharmaceuticals Ltd. (CH) 2010-02-17 EP disclosed
WO-2008132679-A1 BRIDGED SIX-MEMBERED RING COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2008-11-06 WO disclosed