SCHEMBL3662766

SCHEMBL3662766

COc1cc(Nc2ncc3c(n2)C(N2CCOCC2)CCC3)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKMYT1 Q99640 1/20 0.39
CCNT1 O60563 2/20 0.39
CDK9 P50750 2/20 0.39
CDK2 P24941 2/20 0.38
CDK1 P06493 1/20 0.38
CDK4 P11802 1/20 0.38
CCNB1 P14635 1/20 0.38
CCND1 P24385 1/20 0.38
CCNE1 P24864 1/20 0.38
JAK2 O60674 1/20 0.37
ZAP70 P43403 1/20 0.37
SYK P43405 1/20 0.37
IMPDH2 P12268 2/20 0.37
FGFR1 P11362 2/20 0.37
FGFR4 P22455 2/20 0.37
KDR P35968 2/20 0.37
PSEN1 P49768 3/20 0.37
PSEN2 P49810 3/20 0.37
APH1B Q8WW43 3/20 0.37
NCSTN Q92542 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3664634 0.94 PSEN1 (0.39) CDK2CDK1CDK4CCNB1CCND1
SCHEMBL3663912 0.93 PSEN1 (0.40) CDK2CDK1CDK4CCNB1CCND1
SCHEMBL3661445 0.87 LRRK2 (0.40) PKMYT1CCNT1CDK9CDK2CDK1
SCHEMBL3665907 0.84 PLK1 (0.39) CDK2KDRPSEN1PSEN2APH1B
SCHEMBL3657821 0.84 PLK1 (0.39) CDK2KDRPSEN1PSEN2APH1B
SCHEMBL3665261 0.83 PLK1 (0.38) CDK2CDK4CCND1KDRPSEN1
SCHEMBL3661161 0.82 PLK1 (0.38) CDK2CDK1CCNB1KDRPSEN1
SCHEMBL1617106 0.82 PSEN1 (0.56) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3662116 0.81 PDGFRB (0.39) CDK4CCND1KDRPSEN1PSEN2
SCHEMBL3663840 0.81 PSEN1 (0.50) CDK2KDRPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231629-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-09-29 EP disclosed
WO-2009087127-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-07-16 WO disclosed