SCHEMBL366279

SCHEMBL366279

O=Cc1ccccc1OCCN1CCNC1=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
ALDH1A1 P00352 6/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
HPGD P15428 1/20 0.54
HTT P42858 1/20 0.54
RAD52 P43351 1/20 0.46
SCN9A Q15858 3/20 0.45
SCN5A Q14524 2/20 0.45
SCN2A Q99250 1/20 0.45
SCN3A Q9NY46 1/20 0.45
SCN8A Q9UQD0 1/20 0.45
PDK2 Q15119 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.43
POLB P06746 2/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10031750 0.84 HPGD (0.47) MEN1KMT2AALDH1A1SMN1; SMN2HPGD
SCHEMBL365952 0.84 HPGD (0.47) MEN1KMT2AALDH1A1SMN1; SMN2HPGD
SCHEMBL371151 0.84 HPGD (0.47) MEN1KMT2AALDH1A1SMN1; SMN2HPGD
SCHEMBL2563726 0.84 NPC1 (0.50) MEN1KMT2AALDH1A1SMN1; SMN2SCN9A
SCHEMBL2560274 0.82 KDM4E (0.50) MEN1KMT2AALDH1A1SCN9ASCN5A
SCHEMBL15332183 0.81 ALDH1A1 (0.49) MEN1KMT2AALDH1A1SMN1; SMN2SCN9A
SCHEMBL2564218 0.81 KMT2A (0.43) MEN1KMT2AALDH1A1SMN1; SMN2HTT
SCHEMBL19314030 0.81 KMT2A (0.45) MEN1KMT2AALDH1A1SMN1; SMN2HPGD
SCHEMBL18758160 0.80 KMT2A (0.43) MEN1KMT2AALDH1A1SMN1; SMN2SCN9A
SCHEMBL18758195 0.80 MEN1 (0.43) MEN1KMT2AALDH1A1SMN1; SMN2RAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3313823-B1 METHOD FOR SYNTHESIZING MOLECULES HAVING A NITRILE OXIDE FUNCTION MICHELIN & CIE (FR) 2022-11-09 EP disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
EP-3313822-A1 METHOD FOR SYNTHESIZING AROMATIC OXIMES Compagnie Générale des Etablissements Michelin (FR) 2018-05-02 EP disclosed
EP-3313823-A1 METHOD FOR SYNTHESIZING MOLECULES HAVING A NITRILE OXIDE FUNCTION Compagnie Générale des Etablissements Michelin (FR) 2018-05-02 EP disclosed
EP-2593437-B1 MOLECULES HAVING COMBINABLE GROUPS ARKEMA FRANCE (FR) 2017-09-06 EP disclosed
EP-2593437-B1 MOLECULES HAVING COMBINABLE GROUPS ARKEMA FRANCE (FR) 2017-09-06 EP disclosed
WO-2017064296-A1 METHOD FOR SYNTHESISING AROMATIC NITRONES ARKEMA FRANCE (FR) 2017-04-20 WO disclosed
WO-2016207261-A1 METHOD FOR SYNTHESIZING AROMATIC OXIMES COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2016-12-29 WO disclosed
US-20130131279-A1 GRAFT POLYMER TO WHICH COMBINED NITROGEN MOLECULES ARE GRAFTED Mchelin Recherche et Technique S.A. (CH) 2013-05-23 US disclosed
US-20130131279-A1 GRAFT POLYMER TO WHICH COMBINED NITROGEN MOLECULES ARE GRAFTED Mchelin Recherche et Technique S.A. (CH) 2013-05-23 US disclosed
EP-2593485-A1 GRAFT POLYMER TO WHICH COMBINED NITROGEN MOLECULES ARE GRAFTED Compagnie Générale des Etablissements Michelin (FR) 2013-05-22 EP disclosed
EP-2593437-A1 MOLECULES HAVING COMBINABLE GROUPS Arkema France (FR) 2013-05-22 EP disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2012007441-A1 GRAFT POLYMER TO WHICH COMBINED NITROGEN MOLECULES ARE GRAFTED SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2012-01-19 WO disclosed
WO-2012007441-A1 GRAFT POLYMER TO WHICH COMBINED NITROGEN MOLECULES ARE GRAFTED SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2012-01-19 WO disclosed
WO-2012007684-A1 MOLECULES HAVING COMBINABLE GROUPS ARKEMA FRANCE (FR) 2012-01-19 WO disclosed
WO-2012007684-A1 MOLECULES HAVING COMBINABLE GROUPS ARKEMA FRANCE (FR) 2012-01-19 WO disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed