SCHEMBL3662939

SCHEMBL3662939

CC(C)CC1c2ccc(I)cc2CCCN1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 16/20 0.41
MTNR1A P48039 2/20 0.35
AKR1C3 P42330 1/20 0.35
SRD5A1 P18405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639209 0.86 MTNR1B (0.41) MTNR1BMTNR1A
SCHEMBL3664188 0.83 MTNR1B (0.39) MTNR1BAKR1C3
SCHEMBL3657289 0.80 MTNR1B (0.37) MTNR1BMTNR1A
SCHEMBL4032581 0.79 MTNR1B (0.48) MTNR1BMTNR1A
SCHEMBL2123940 0.78 MTNR1B (0.47) MTNR1BMTNR1A
SCHEMBL3664253 0.78 MTNR1B (0.47) MTNR1BMTNR1A
SCHEMBL4638202 0.77 MTNR1B (0.35) MTNR1BMTNR1A
SCHEMBL2984099 0.77 DPP4 (0.38) AKR1C3SRD5A1
SCHEMBL2123210 0.75 MTNR1B (0.45) MTNR1BMTNR1AAKR1C3
SCHEMBL2123219 0.73 MTNR1B (0.43) MTNR1BMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222669-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (SIP) Glaxo Group Limited (GB) 2010-09-01 EP disclosed
WO-2009080725-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (SIP) GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed