SCHEMBL3663738

SCHEMBL3663738

CC(C)(C)C[C@@H](c1ccc(Br)cc1)N(CCC(=NSC(C)(C)C)c1ccccc1)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3655180 0.78 ALDH1A1 (0.35) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL3768894 0.78 ALDH1A1 (0.35) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL3768901 0.78 ALDH1A1 (0.35) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL3663740 0.74 ALDH1A1 (0.38) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL1464059 0.73 RIPK1 (0.43) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1464039 0.68 IGF1R (0.36) ALDH1A1MAPTMEN1KMT2A
SCHEMBL3661629 0.65 NPC1 (0.44) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL3661631 0.65 NPC1 (0.44) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL3207998 0.63 ALDH1A1 (0.35) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL3207967 0.63 ALDH1A1 (0.35) KDM4EALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220052-B1 CYCLIC UREA INHIBITORS OF 11ß-HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS INC (US) 2015-03-25 EP disclosed
EP-2220052-A1 CYCLIC UREA INHIBITORS OF 11 -HYDROXYSTEROID DEHYDROGENASE 1 Vitae Pharmaceuticals, Inc. (US) 2010-08-25 EP disclosed
WO-2009061498-A1 CYCLIC UREA INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-05-14 WO disclosed