SCHEMBL3663816

SCHEMBL3663816

NC(=O)c1cccc(-c2ccc3cc[nH]c3c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.58
CCND1 P24385 1/20 0.58
CCNC P24863 1/20 0.58
CDK8 P49336 1/20 0.58
CDK7 P50613 1/20 0.58
CDK9 P50750 1/20 0.58
CCNH P51946 1/20 0.58
MNAT1 P51948 1/20 0.58
CDK6 Q00534 1/20 0.58
LCK P06239 1/20 0.52
BTK Q06187 1/20 0.52
GHSR Q92847 3/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
ENPP2 Q13822 1/20 0.50
HSD17B10 Q99714 1/20 0.50
ERN1 O75460 2/20 0.49
TDP2 O95551 1/20 0.49
AAK1 Q2M2I8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL982808 0.88 CCNT1 (0.62) CCNT1CCND1CCNCCDK8CDK7
SCHEMBL2277469 0.86 KDM4E (0.70) GHSRKDM4EALDH1A1HPGDENPP2
Benzene SCHEMBL27399226 0.83 ALDH1A1 (0.71) CCNT1CCND1CCNCCDK8CDK7
SCHEMBL30201702 0.83 ALDH1A1 (0.70) LCKGHSRKDM4EALDH1A1HPGD
SCHEMBL50552 0.83 ALDH1A1 (0.70) LCKGHSRKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL8915608 0.82 ALDH1A1 (0.68) LCKGHSRKDM4EALDH1A1HPGD
SCHEMBL29566955 0.82 ALDH1A1 (0.68) LCKGHSRKDM4EALDH1A1HPGD
Iodide SCHEMBL8916427 0.82 ALDH1A1 (0.68) LCKGHSRKDM4EALDH1A1HPGD
Bromide SCHEMBL8916350 0.82 ALDH1A1 (0.68) LCKGHSRKDM4EALDH1A1HPGD
SCHEMBL1513161 0.81 CDK8 (0.62) CDK8GHSRERN1PLAUPLAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8642788-B2 Activators of executioner procaspases 3, 6 and 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-02-04 US disclosed
CN-101965189-A Activators of pro-caspase 3, 6 and 7 UNIV CALIFORNIA 2011-02-02 CN disclosed
EP-2237784-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 The Regents of the University of California (US) 2010-10-13 EP disclosed
WO-2009089508-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-07-16 WO disclosed