SCHEMBL3664867

SCHEMBL3664867

O=C(O)C1CCOC(c2ccc(-c3ccccc3)cc2)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.54
NPC1 O15118 2/20 0.54
AKR1C3 P42330 1/20 0.45
AKR1C1 Q04828 1/20 0.45
KDM1A O60341 4/20 0.41
MAOB P27338 1/20 0.41
FFAR1 O14842 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
DGAT1 O75907 1/20 0.39
LTA4H P09960 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
EPHX1 P07099 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3859730 0.91 AKR1C3 (0.54) RAB9ANPC1AKR1C3AKR1C1FFAR1
SCHEMBL29428983 0.83 NOTUM (0.41) AKR1C3AKR1C1KDM1ALTA4HMEN1
SCHEMBL12477256 0.83 AKR1C3 (0.39) RAB9ANPC1AKR1C3AKR1C1KDM1A
SCHEMBL2077447 0.79 GAA (0.45) RAB9ANPC1KDM1AMAOBMEN1
SCHEMBL9940281 0.78 TSHR (0.41) AKR1C3AKR1C1KDM1ALTA4HKMT2A
SCHEMBL29705664 0.77 FFAR1 (0.47) RAB9ANPC1KDM1AMAOBFFAR1
SCHEMBL4618863 0.75 KDM1A (0.43) AKR1C3AKR1C1KDM1AFFAR1HPGD
SCHEMBL29428973 0.75 AKR1C3 (0.42) NPC1AKR1C3AKR1C1CYP1A2CYP2C9
SCHEMBL29428980 0.75 AKR1C3 (0.41) AKR1C3AKR1C1KDM1AMEN1KMT2A
Biphenyl SCHEMBL7614586 0.74 RAB9A (0.63) RAB9ANPC1AKR1C3AKR1C1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2142505-A1 SULFONAMIDES AND PHARMACEUTICAL COMPOSITIONS THEREOF Pfizer, Inc. (US) 2010-01-13 EP disclosed
WO-2008120093-A1 SULFONAMIDES AND PHARMACEUTICAL COMPOSITIONS THEREOF PFIZER INC. (US) 2008-10-09 WO disclosed