SCHEMBL3665733

SCHEMBL3665733

CC(C)(C)Nc1cc(-c2cncc(-c3ccc(N4CCNCC4)cc3)c2)cc(-c2ccccn2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.49
ACVR1 Q04771 7/20 0.48
ACVR1B P36896 1/20 0.48
HTR1A P08908 1/20 0.45
HTR7 P34969 1/20 0.45
PIM1 P11309 2/20 0.45
PIM3 Q86V86 2/20 0.45
KARS1 Q15046 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
CHEK1 O14757 3/20 0.40
ACVRL1 P37023 2/20 0.40
CDK7 P50613 1/20 0.39
RIPK2 O43353 1/20 0.39
NOD2 Q9HC29 1/20 0.39
FLT3 P36888 1/20 0.38
TYRO3 Q06418 1/20 0.38
MERTK Q12866 1/20 0.38
GAS6 Q14393 1/20 0.38
PIM2 Q9P1W9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3725771 0.85 CCNC (0.53)
SCHEMBL3718900 0.79 GPR39 (0.44) TGFBR1PIM1FLT3
SCHEMBL3727190 0.79 CHEK1 (0.48) ACVR1CHEK1
SCHEMBL3667875 0.78 GPR39 (0.37)
SCHEMBL3727963 0.76 ABL1 (0.50) TYRO3MERTK
SCHEMBL3723126 0.76 PIK3CD (0.40) TGFBR1ACVR1HDAC1
SCHEMBL3725755 0.76 ABL1 (0.48) TGFBR1CHEK1
SCHEMBL3666866 0.75 ADORA3 (0.45) TGFBR1
SCHEMBL3726132 0.74 ABL1 (0.48) PIM1
SCHEMBL3718285 0.74 CCNC (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242742-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2010-10-27 EP disclosed
WO-2009087212-A2 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2009-07-16 WO disclosed