SCHEMBL3666055

SCHEMBL3666055

C=C(c1cccc(OC)c1)c1ccc2c(c1)c1c(C(=C)c3cccc(OC)c3)ccnc1n2S(=O)(=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
HSD11B1 P28845 1/20 0.39
HTR6 P50406 9/20 0.38
KAT6A Q92794 1/20 0.37
MAPK1 P28482 1/20 0.37
ELANE P08246 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL675269 0.90 HDAC3 (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3671977 0.90 SRC (0.37) HTR6PTGDR2
SCHEMBL676947 0.85 PTGDR2 (0.40) HTR6KAT6APOLBL3MBTL1PTGDR2
SCHEMBL674879 0.83 PTGDR2 (0.37) HTR6KAT6APTGDR2
SCHEMBL675869 0.81 HTR6 (0.40) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3665214 0.81 HDAC3 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL676361 0.80 HDAC3 (0.41) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL675466 0.79 ENPP3 (0.38) HTR6PTGDR2
SCHEMBL675759 0.74 PTGDR2 (0.37) HTR6MAPK1PTGDR2
SCHEMBL16241827 0.73 HTR6 (0.41) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed