SCHEMBL3666221

SCHEMBL3666221

Cn1c(CN(CCCN2CCC(n3c(=O)[nH]c4ccccc43)CC2)Cc2ccccc2)cc2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.57
CYP2C9 P11712 1/20 0.57
CHRM1 P11229 4/20 0.55
PMP22 Q01453 3/20 0.55
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
NPSR1 Q6W5P4 2/20 0.55
OPRM1 P35372 7/20 0.54
OPRK1 P41145 3/20 0.54
OPRL1 P41146 2/20 0.54
BCHE P06276 1/20 0.53
ACHE P22303 1/20 0.53
ADRA1A P35348 3/20 0.52
ADRA1D P25100 2/20 0.52
ADRA1B P35368 1/20 0.52
DRD2 P14416 4/20 0.51
KCNH2 Q12809 4/20 0.51
HTR1A P08908 3/20 0.51
HTR2A P28223 3/20 0.51
DRD3 P35462 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3746351 0.89 CYP2D6 (0.67) CYP2D6CYP2C9CHRM1PMP22KDM4E
SCHEMBL3745582 0.86 CHRM1 (0.67) CYP2D6CYP2C9CHRM1PMP22KDM4E
SCHEMBL1835801 0.86 CHRM1 (0.53) CYP2D6CYP2C9CHRM1PMP22KDM4E
Hydrochloric Acid SCHEMBL1836997 0.85 CHRM1 (0.52) CYP2D6CYP2C9CHRM1PMP22KDM4E
SCHEMBL3636721 0.84 CHRM1 (0.54) CHRM1PMP22KDM4EALDH1A1NPSR1
SCHEMBL1835330 0.84 KDM4E (0.43) CYP2D6CYP2C9CHRM1PMP22KDM4E
SCHEMBL3635266 0.83 OPRM1 (0.69) CYP2D6CYP2C9CHRM1PMP22KDM4E
SCHEMBL3665754 0.82 CYP2D6 (0.57) CYP2D6CYP2C9CHRM1PMP22KDM4E
SCHEMBL1835328 0.79 BCHE (0.38) CYP2D6CYP2C9CHRM1PMP22KDM4E
SCHEMBL3806337 0.78 OPRM1 (0.70) CYP2D6CYP2C9CHRM1PMP22OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155676-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS Commissariat à l'Energie Atomique (FR) 2010-02-24 EP claimed
WO-2008146172-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-12-04 WO claimed