SCHEMBL3669767

SCHEMBL3669767

Cn1c(CN(CC[C@H]2CC(n3c(=O)[nH]c4ccccc43)CCN2C(=O)O)Cc2ccccc2)cc2ccccc21.O=C(O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1CCCN(Cc1ccccc1)Cc1ccnc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
TNKS O95271 2/20 0.37
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
PLD2 O14939 2/20 0.37
PLD1 Q13393 2/20 0.37
TACR1 P25103 4/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PMP22 Q01453 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
AKT1 P31749 3/20 0.36
ABL1 P00519 1/20 0.34
RIN1 Q13671 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
AKT2 P31751 1/20 0.34
AKT3 Q9Y243 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400388 0.91 TNKS (0.42) BCHEACHETNKSPARP1PARP2
SCHEMBL1838933 0.91 TNKS (0.42) BCHEACHETNKSPARP1PARP2
SCHEMBL1835330 0.90 KDM4E (0.43) BCHEACHEPLD2PLD1KDM4E
SCHEMBL1835697 0.89 OPRM1 (0.42) BCHEACHETNKSPARP1PARP2
SCHEMBL1838230 0.88 TNKS (0.44) BCHEACHETNKSPARP1PARP2
SCHEMBL3403019 0.83 CYP3A4 (0.43) BCHEACHETNKSPARP1PARP2
SCHEMBL1834696 0.82 OPRM1 (0.41) BCHEACHETNKSPARP1PARP2
SCHEMBL3806376 0.82 CYP3A4 (0.44) BCHEACHETNKSPARP1PARP2
SCHEMBL1835272 0.81 OPRM1 (0.50) BCHEACHEPLD2PLD1KDM4E
SCHEMBL3403017 0.81 OPRM1 (0.50) BCHEACHEPLD2PLD1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155676-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS Commissariat à l'Energie Atomique (FR) 2010-02-24 EP disclosed
WO-2008146172-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-12-04 WO disclosed