SCHEMBL3669946

SCHEMBL3669946

Fc1ccc(Br)cc1-c1nc(NCCNc2ccccn2)c2nccnc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.44
PRKD3 O94806 1/20 0.44
PRKD1 Q15139 1/20 0.44
PRKD2 Q9BZL6 1/20 0.44
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
METAP1 P53582 4/20 0.34
CYP1A2 P05177 1/20 0.34
ADRA1A P35348 2/20 0.33
HTR1A P08908 1/20 0.33
CYP2C19 P33261 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
PIP4K2C Q8TBX8 1/20 0.32
METAP2 P50579 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2128108 0.84 TGFBR1 (0.48) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL2126398 0.78 TGFBR1 (0.64) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL2126260 0.75 TGFBR1 (0.51) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL2128085 0.74 TGFBR1 (0.77) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL2125422 0.71 TGFBR1 (0.50) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL2128905 0.71 TGFBR1 (0.59) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL2127268 0.70 ALDH1A1 (0.41) MEN1MAPTKMT2A
SCHEMBL2128877 0.69 TGFBR1 (0.54) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL27732302 0.69 TGFBR1 (0.42) TGFBR1PRKD3PRKD1PRKD2FLT1
SCHEMBL2127625 0.68 MEN1 (0.38) TGFBR1PRKD3PRKD1PRKD2FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881834-B1 PTERIDINES USEFUL AS HCV INHIBITORS AND METHODS FOR THE PREPARATION THEREOF JANSSEN R & D IRELAND (IE) 2012-04-25 EP disclosed