SCHEMBL3670277

SCHEMBL3670277

COc1ccc(N)c(Nc2ccc3c(c2)CCC(N(C(=O)O)C(c2cc4c(cn2)OCCO4)C(C)(C)C)C3)n1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.32
WEE1 P30291 1/20 0.32
CSF1R P07333 1/20 0.32
CDK4 P11802 1/20 0.32
CDK6 Q00534 1/20 0.32
SYK P43405 3/20 0.31
BACE1 P56817 2/20 0.31
BACE2 Q9Y5Z0 2/20 0.31
PIK3CA P42336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3668331 0.83 TSHR (0.31) KCNH2
SCHEMBL3025535 0.82 KCNH2 (0.39) KCNH2
SCHEMBL3020658 0.79 TSHR (0.31) KCNH2
SCHEMBL3666201 0.79 TSHR (0.31) KCNH2
SCHEMBL3016694 0.72 KCNH2 (0.37) KCNH2
SCHEMBL3016687 0.72 KCNH2 (0.37) KCNH2
SCHEMBL3669003 0.71 KCNH2 (0.35) KCNH2
SCHEMBL3013394 0.68 KCNH2 (0.34) KCNH2SYK
SCHEMBL3149928 0.67 KCNH2 (0.40) KCNH2
SCHEMBL3025404 0.63 KDM4C (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139898-A1 COMPOUNDS Glaxo Group Limited (GB) 2010-01-06 EP disclosed
WO-2008128961-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-10-30 WO disclosed