SCHEMBL3668331

SCHEMBL3668331

CC(C)(C)C(c1cc2c(cn1)OCCO2)N(C(=O)O)C1CCc2cc(N)ccc2C1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.31
HTR2C P28335 1/20 0.31
KCNH2 Q12809 1/20 0.31
MCHR1 Q99705 1/20 0.31
NR1H2 P55055 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3666201 0.90 TSHR (0.31) TSHRHTR2CKCNH2MCHR1
SCHEMBL3020658 0.90 TSHR (0.31) TSHRHTR2CKCNH2MCHR1
SCHEMBL3670277 0.83 KCNH2 (0.32) KCNH2
SCHEMBL3013221 0.75 MCHR1 (0.35) HTR2CKCNH2MCHR1
SCHEMBL3666877 0.73 NR1H2 (0.34) HTR2CKCNH2MCHR1NR1H2
SCHEMBL3028019 0.64 MCHR1 (0.35) HTR2CKCNH2MCHR1
SCHEMBL3020655 0.63 MCHR1 (0.34) HTR2CKCNH2MCHR1
SCHEMBL8145781 0.62 DRD3 (0.41)
SCHEMBL8145785 0.62 DRD3 (0.41)
SCHEMBL3468089 0.61 DRD2 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139898-A1 COMPOUNDS Glaxo Group Limited (GB) 2010-01-06 EP disclosed
WO-2008128961-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-10-30 WO disclosed