SCHEMBL3670338

SCHEMBL3670338

Clc1cccc(C(c2cccnc2)c2cnc[nH]2)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 2/20 0.44
CYP19A1 P11511 1/20 0.43
SLC6A2 P23975 5/20 0.41
SLC6A4 P31645 4/20 0.41
SLC6A3 Q01959 4/20 0.41
CFTR P13569 1/20 0.41
GOPC Q9HD26 1/20 0.41
CYP2D6 P10635 3/20 0.40
KCNH2 Q12809 3/20 0.40
HRH3 Q9Y5N1 2/20 0.39
HRH4 Q9H3N8 1/20 0.39
ADRA2A P08913 8/20 0.39
ADRA2B P18089 8/20 0.39
ADRA2C P18825 8/20 0.39
ADRA1A P35348 7/20 0.39
ADRA1B P35368 6/20 0.39
ADRA1D P25100 5/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1638483 0.88 ADRA2A (0.43) CYP19A1SLC6A2CYP2D6KCNH2ADRA2A
SCHEMBL3062595 0.87 CYP19A1 (0.41) KCNA5CYP19A1SLC6A2SLC6A4SLC6A3
SCHEMBL3062592 0.86 ADRA2A (0.40) CYP19A1SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL13089104 0.80 KCNA5 (0.45) KCNA5CYP19A1SLC6A2SLC6A4SLC6A3
SCHEMBL13247022 0.79 CYP19A1 (0.39) KCNA5CYP19A1SLC6A2SLC6A4SLC6A3
SCHEMBL3063952 0.79 HRH3 (0.41) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL3064587 0.79 ADRA2A (0.62) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL3061266 0.79 ADRA2A (0.41) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL3060612 0.78 SLC6A2 (0.46) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL3061486 0.78 GAA (0.55) CYP19A1SLC6A2SLC6A4SLC6A3CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101743240-B ((phenyl) imidazolyl) methyl heteroaryl compounds ALLERGAN INC 2013-07-17 CN disclosed
EP-2155715-B1 ((PHENYL)IMIDAZOLYL)METHYLHETEROARYL COMPOUNDS ALLERGAN INC (US) 2013-03-13 EP disclosed
EP-2155715-A1 ((PHENYL)IMIDAZOLYL)METHYLHETEROARYL COMPOUNDS ALLERGAN, INC. (US) 2010-02-24 EP disclosed
WO-2008141312-A1 ((PHENYL)IMIDAZOLYL)METHYLHETEROARYL COMPOUNDS ALLERGAN, INC. (US) 2008-11-20 WO disclosed