SCHEMBL3670923

SCHEMBL3670923

O=[N+]([O-])c1cc(F)c(F)nc1NC(CO)c1ccc(F)cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 3/20 0.36
KCNH2 Q12809 2/20 0.36
TDP1 Q9NUW8 2/20 0.33
ATM Q13315 1/20 0.33
TRPV3 Q8NET8 1/20 0.32
PRKCQ Q04759 2/20 0.32
MEN1 O00255 2/20 0.31
LMNA P02545 2/20 0.31
KMT2A Q03164 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
ALDH1A1 P00352 2/20 0.31
CA1 P00915 1/20 0.31
MMP2 P08253 1/20 0.31
CA14 Q9ULX7 1/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
PKM P14618 1/20 0.31
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3008853 1.00 NTRK1 (0.36) NTRK1KCNH2TDP1ATMTRPV3
SCHEMBL2570152 0.84 ADRB2 (0.37) NTRK1TDP1ATMMEN1LMNA
SCHEMBL3136036 0.84 ADRB2 (0.37) NTRK1TDP1ATMMEN1LMNA
SCHEMBL2570151 0.84 ADRB2 (0.37) NTRK1TDP1ATMMEN1LMNA
SCHEMBL3009495 0.83 JAK3 (0.42) NTRK1KCNH2PRKCQ
SCHEMBL3671586 0.83 JAK3 (0.42) NTRK1KCNH2PRKCQ
SCHEMBL3018456 0.81 JAK3 (0.54) NTRK1
SCHEMBL3024160 0.79 NTRK1 (0.42) NTRK1KCNH2
SCHEMBL3012333 0.78 NTRK1 (0.43) NTRK1KCNH2
SCHEMBL3008289 0.77 NTRK1 (0.44) NTRK1KCNH2PRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155742-A1 5-AMINOPYRAZOL-3-YL-3H-IMIDAZO [4,5-B]PYRIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF CANCER AstraZeneca AB (SE) 2010-02-24 EP disclosed
WO-2008129255-A1 5-AMINOPYRAZOL-3-YL-3H-IMIDAZO [4,5-B] PYRIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-10-30 WO disclosed