SCHEMBL367125

SCHEMBL367125

NC(O)c1ccncc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27503629 0.77 SLC6A2 (0.48)
SCHEMBL7680971 0.77 CYP3A4 (0.67)
SCHEMBL20710609 0.77 CYP3A4 (0.48)
SCHEMBL2081194 0.77
SCHEMBL2639851 0.77
SCHEMBL16781699 0.77 DPP4 (0.50)
SCHEMBL1892118 0.77 CYP3A4 (0.48)
SCHEMBL3851200 0.74 TAAR1 (0.60)
SCHEMBL387892 0.72
SCHEMBL1515379 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248425-B Two-dimensional Ag (I) complex synthesized based on silver hexafluorophosphate as well as synthesis method and application thereof 天津师范大学 2022-11-08 CN claimed
CN-113248526-B Two-dimensional Ag (I) complex synthesized based on silver trifluoroacetate and synthesis method and application thereof 天津师范大学 2022-05-31 CN claimed
CN-113248527-B Three-dimensional Ag (I) complex synthesized based on silver methylsulfonate and synthesis method and application thereof 天津师范大学 2022-05-31 CN claimed
CN-113248528-B Three-dimensional Ag (I) complex synthesized based on silver hexafluorosilicate and synthesis method and application thereof 天津师范大学 2022-05-31 CN claimed
CN-113248526-B Two-dimensional Ag (I) complex synthesized based on silver trifluoroacetate and synthesis method and application thereof 天津师范大学 2022-05-31 CN disclosed
CN-113248528-B Three-dimensional Ag (I) complex synthesized based on silver hexafluorosilicate and synthesis method and application thereof 天津师范大学 2022-05-31 CN disclosed
CN-113248527-B Three-dimensional Ag (I) complex synthesized based on silver methylsulfonate and synthesis method and application thereof 天津师范大学 2022-05-31 CN disclosed
CN-104854091-B The amine derivative of 5 fluorine N (base of pyridine 2) pyridine 2 containing sulfone group 拜耳药业股份公司 2018-04-03 CN disclosed
CN-105102444-B Sulfomimino-containing 5-fluoro-N- (pyridin-2-yl) pyridin-2-amine derivatives 拜耳医药股份有限公司 2017-08-01 CN disclosed
CN-105283453-A N- (pyridin-2-yl) pyrimidin-4-amine derivatives containing sulfone group Bayer Pharma AG 2016-01-27 CN disclosed
CN-105102444-A Sulfomimino-containing 5-fluoro-N- (pyridin-2-yl) pyridin-2-amine derivatives Bayer Pharma AG 2015-11-25 CN disclosed
CN-104918932-A N-(pyridin-2-yl)pyrimidin-4-amine derivatives containing a sulfoximine group Bayer Pharma AG 2015-09-16 CN disclosed
CN-104854091-A 5-fluoro-n-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group Bayer Pharma AG 2015-08-19 CN disclosed
EP-2578579-A1 Benzothiophene carboxamide compounds, composition and applications thereof National Institute of Immunology (IN) 2013-04-10 EP disclosed
US-20120016014-A1 BENZOTHIOPHENE CARBOXAMIDE COMPOUNDS, COMPOSITION AND APPLICATIONS THEREOF INDIAN INSTITUTE OF SCIENCE (IN) 2012-01-19 US disclosed
US-3953463-A 2-Aryl-6-trifluoromethyl-4-pyridyl-carbinolamine antimalarials THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1976-04-27 US disclosed
US-3940404-A PLASMODIAL INFECTIONS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1976-02-24 US disclosed
US-3886167-A 2-Aryl-6-trifluoromethyl-4-pyridylcarbinolamine antimalarials US ARMY 1975-05-27 US disclosed
US-3764604-A 4-PYRIDYLCARBINOLAMINE ANTI-MALARIALS US ARMY 1973-10-09 US disclosed