SCHEMBL3671608

SCHEMBL3671608

CC1C[C@H]2CN[C@H](CNC(=O)c3snc4ccccc34)[C@H]2C1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SSTR4 P31391 8/20 0.33
GBA1 P04062 1/20 0.31
SSTR1 P30872 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL496230 0.82 MAPT (0.43)
SCHEMBL2445362 0.82 MAPT (0.43)
SCHEMBL3668373 0.80 ROCK1 (0.35) KDM4EALDH1A1HPGDHTTHSD17B10
SCHEMBL496329 0.76 HIF1A (0.43) SSTR4
SCHEMBL496213 0.76 CYP3A4 (0.47) KDM4EALDH1A1MAPK1HSD17B10SSTR4
SCHEMBL3641052 0.74 ACKR3 (0.36) KDM4EALDH1A1HPGDMAPK1HTT
SCHEMBL496447 0.68 HTR4 (0.48)
SCHEMBL496485 0.67 KDM4E (0.34) KDM4EALDH1A1HPGDHTTHSD17B10
SCHEMBL8209794 0.67 MAPT (0.50) KDM4EALDH1A1HTTHSD17B10
SCHEMBL2450556 0.67 HCRTR1 (0.45) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164847-A1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS Actelion Pharmaceuticals Ltd. (CH) 2010-03-24 EP disclosed
WO-2009004584-A1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2009-01-08 WO disclosed