SCHEMBL3671654

SCHEMBL3671654

c1coc(-c2ccc3[nH]c4nccc(-c5ccco5)c4c3c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.46
CDK1 P06493 1/20 0.46
CCNB1 P14635 1/20 0.46
GSK3B P49841 1/20 0.46
CDK5 Q00535 1/20 0.46
CDK5R1 Q15078 1/20 0.46
CCNB3 Q8WWL7 1/20 0.46
ALK Q9UM73 11/20 0.46
GABRA1 P14867 2/20 0.45
GABRG2 P18507 2/20 0.45
GABRB3 P28472 2/20 0.45
GABRA5 P31644 2/20 0.45
GABRA3 P34903 2/20 0.45
GABRA2 P47869 2/20 0.45
GABRA6 Q16445 2/20 0.45
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
GABRA4 P48169 1/20 0.43
EGFR P00533 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL676261 0.85 ALK (0.52) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL668576 0.83 ALK (0.47) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL3723800 0.78 CNR2 (0.43) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL31318484 0.77 GABRA1 (0.55) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL677069 0.77 GABRA1 (0.39) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL676503 0.75 GABRA1 (0.49) ALKGABRA1GABRG2GABRB3GABRA5
SCHEMBL675430 0.74 ALK (0.70) ALKMAPK14
SCHEMBL677068 0.74 CNR2 (0.39) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL676627 0.74 ALK (0.45) ALKGABRA1GABRG2GABRB3GABRA5
SCHEMBL676628 0.74 ALK (0.45) ALKGABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed