SCHEMBL3671916

SCHEMBL3671916

O=c1[nH]c2ccccc2n1C1CCN(CCOCc2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 5/20 0.72
DRD2 P14416 5/20 0.72
KCNH2 Q12809 5/20 0.72
OPRM1 P35372 8/20 0.69
OPRK1 P41145 3/20 0.69
OPRL1 P41146 1/20 0.69
CYP2D6 P10635 3/20 0.67
CYP2C9 P11712 1/20 0.67
PMP22 Q01453 3/20 0.64
KDM4E B2RXH2 2/20 0.64
ALDH1A1 P00352 2/20 0.64
NPSR1 Q6W5P4 2/20 0.64
HTR1A P08908 3/20 0.63
HTR2A P28223 3/20 0.63
DRD3 P35462 3/20 0.63
CHRM5 P08912 2/20 0.63
CHRM2 P08172 2/20 0.62
CHRM4 P08173 1/20 0.62
CHRM3 P20309 1/20 0.62
ADRA1A P35348 3/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24709114 0.85 CYP2D6 (0.74) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL31000422 0.85 CYP2D6 (0.74) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL5777954 0.85 OPRM1 (0.77) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL5984495 0.84 CYP2D6 (0.85) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL2993173 0.84 CYP2D6 (0.73) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL2982735 0.84 CHRM1 (0.71) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL6404540 0.84 PLD1 (0.81) CHRM1DRD2KCNH2OPRM1OPRK1
Oxiperomide SCHEMBL123291 0.84 CHRM1 (1.00) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL24708725 0.84 CHRM1 (0.73) CHRM1DRD2KCNH2OPRM1OPRK1
SCHEMBL5773820 0.84 CHRM1 (0.75) CHRM1DRD2KCNH2OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155676-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS Commissariat à l'Energie Atomique (FR) 2010-02-24 EP claimed
WO-2008146172-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-12-04 WO claimed