SCHEMBL367400

SCHEMBL367400

CC1(C)c2cc(Br)ccc2-c2ccc(-c3ccc(-c4ccc5ccccc5c4)cc3)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.47
LPL P06858 1/20 0.43
LIPG Q9Y5X9 1/20 0.43
ESR1 P03372 2/20 0.42
ESR2 Q92731 2/20 0.42
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
GSTP1 P09211 1/20 0.39
PDK2 Q15119 3/20 0.38
ALOX5 P09917 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
PTGER3 P43115 2/20 0.36
CYP1A2 P05177 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL429070 0.98 CYP2A6 (0.48) CYP2A6LPLLIPGESR1ESR2
SCHEMBL429952 0.98 CYP2A6 (0.48) CYP2A6LPLLIPGESR1ESR2
SCHEMBL2472869 0.98 CYP2A6 (0.48) CYP2A6LPLLIPGESR1ESR2
SCHEMBL19152839 0.91 CYP2A6 (0.44) CYP2A6LPLLIPGESR1ESR2
SCHEMBL20938291 0.91 CYP11B1 (0.42) CYP2A6LPLLIPGESR1ESR2
SCHEMBL25770839 0.89 CYP2A6 (0.42) CYP2A6LPLLIPGESR1ESR2
SCHEMBL431640 0.88 CYP2A6 (0.43) CYP2A6LPLLIPGCYP11B1CYP11B2
SCHEMBL322802 0.88 CYP2A6 (0.43) CYP2A6LPLLIPGCYP11B1CYP11B2
SCHEMBL431820 0.87 MAPK1 (0.47) PDK2SMN1; SMN2
SCHEMBL429037 0.87 MAPK1 (0.47) PDK2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415752-B1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO (JP) 2016-03-09 EP disclosed
US-9184395-B2 Aromatic amine derivative and organic electroluminescent element using same IDEMITSU KOSAN CO., LTD. (JP) 2015-11-10 US disclosed
US-9184395-B2 Aromatic amine derivative and organic electroluminescent element using same IDEMITSU KOSAN CO., LTD. (JP) 2015-11-10 US disclosed
US-8980442-B2 Aromatic amine derivative and organic electroluminescent element using same MITSUI CHEMICALS, INC. (JP) 2015-03-17 US disclosed
CN-102356060-A Aromatic amine derivative and organic electroluminescent element using same MITSUI CHEMICALS INC 2012-02-15 CN disclosed
EP-2415752-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME Mitsui Chemicals, Inc. (JP) 2012-02-08 EP disclosed
US-20120012832-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME MITSUI CHEMICALS, INC. (JP) 2012-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120012832-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME MAOA, MAOB, TYR CYP2A6 772/4885LPL 1699/4885LIPG 1996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.