SCHEMBL3678664

SCHEMBL3678664

O=C(CC(Sc1ccc(Cl)cc1)C(=O)O)c1ccc(Cl)cc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.80
MAPT P10636 4/20 0.80
LMNA P02545 2/20 0.80
NPSR1 Q6W5P4 2/20 0.80
HSP90AA1 P07900 1/20 0.80
THRB P10828 1/20 0.80
KMT2A Q03164 4/20 0.72
MEN1 O00255 2/20 0.72
BCL2L1 Q07817 1/20 0.72
MCL1 Q07820 1/20 0.72
ATM Q13315 1/20 0.63
POLB P06746 3/20 0.58
HTT P42858 2/20 0.58
RECQL P46063 1/20 0.58
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 2/20 0.54
HSD17B10 Q99714 1/20 0.54
MMP2 P08253 3/20 0.50
MMP3 P08254 3/20 0.50
MMP9 P14780 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL728170 0.94 MAPT (0.71) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL728174 0.94 MAPT (0.71) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL225482 0.93 ALDH1A1 (0.86) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL726525 0.93 KMT2A (0.76) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL727031 0.93 ALDH1A1 (0.86) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL726709 0.89 ALDH1A1 (0.70) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL225008 0.89 ALDH1A1 (1.00) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL728190 0.89 ALDH1A1 (0.70) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL230158 0.87 ALDH1A1 (0.80) ALDH1A1MAPTLMNANPSR1HSP90AA1
SCHEMBL728416 0.86 ALDH1A1 (0.62) ALDH1A1MAPTLMNANPSR1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7727977-B2 Kynurenine 3-hydroxylase inhibitors for the treatment of diabetes MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2010-06-01 US disclosed
US-7727977-B2 Kynurenine 3-hydroxylase inhibitors for the treatment of diabetes MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2010-06-01 US disclosed
US-7727977-B2 Kynurenine 3-hydroxylase inhibitors for the treatment of diabetes MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2010-06-01 US disclosed