SCHEMBL3680346

SCHEMBL3680346

Oc1ccc(C(c2ccc(O)c(-c3ccccc3)c2)(C(F)(F)F)C(F)(F)F)cc1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.52
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
BCL2L1 Q07817 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ESR1 P03372 2/20 0.44
ESR2 Q92731 2/20 0.44
PELI1 Q96FA3 1/20 0.42
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
ALOX5 P09917 2/20 0.41
PTGDR2 Q9Y5Y4 2/20 0.40
PTPN5 P54829 3/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
KIF11 P52732 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
BRD4 O60885 1/20 0.36
NR1I2 O75469 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16429040 0.85 BACE1 (0.56) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL3665838 0.81 BACE1 (0.45) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL28445672 0.80 BACE1 (0.46) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL12191322 0.79 KIF11 (0.39) BACE1ESR1ESR2PTGDR2PTPN5
SCHEMBL136305 0.78 BACE1 (0.56) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL29375340 0.78 BACE1 (0.56) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL29602069 0.78 BACE1 (0.56) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL7916383 0.78 BACE1 (0.56) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL3418225 0.78 BACE1 (0.56) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL23861344 0.76 ESR2 (0.62) BACE1ALDH1A1HPGDBCL2L1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10416581-B2 Electrophotographic photosensitive member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2019-09-17 US disclosed
EP-3062153-B1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, METHOD FOR MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KK (JP) 2018-09-26 EP disclosed
US-20180059558-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2018-03-01 US disclosed
US-9864284-B2 Electrophotographic photosensitive member, method for manufacturing electrophotographic photosensitive member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2018-01-09 US disclosed
US-9753385-B2 Electrophotographic photosensitive member, method for manufacturing electrophotographic photosensitive member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2017-09-05 US disclosed
US-9563139-B2 Electrophotographic photosensitive member, process cartridge and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2017-02-07 US disclosed
US-20160252829-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, METHOD FOR MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-09-01 US disclosed
US-20160252830-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, METHOD FOR MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-09-01 US disclosed
EP-3062153-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, METHOD FOR MANUFACTURING ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS Canon Kabushiki Kaisha (JP) 2016-08-31 EP disclosed
US-20160124328-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-05-05 US disclosed
US-7700714-B2 Optical element and achromatic lens TEIJIN CHEMICALS, LTD. (JP) 2010-04-20 US disclosed
US-20090143560-A1 Optical Element and Achromatic Lens TEIJIN CHEMICALS, LTD. 2009-06-04 US disclosed
EP-1947131-A1 OPTICAL DEVICE AND ACHROMATIC LENS Teijin Chemicals, Ltd. (JP) 2008-07-23 EP disclosed
US-6258498-B1 POLYCARBONATE PROTECTIVE COATING CANON KABUSHIKI KAISHA (JP) 2001-07-10 US disclosed