SCHEMBL3684008

SCHEMBL3684008

C=CC(C)(C)c1ccc(OC)c(C=CC(=O)c2ccc(NCCCN(C)C)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 11/20 0.48
ABCG2 Q9UNQ0 2/20 0.47
IDH1 O75874 1/20 0.47
ABCB1 P08183 1/20 0.47
UGT1A1 P22309 1/20 0.47
DPP4 P27487 1/20 0.47
ABCC1 P33527 1/20 0.47
PRMT6 Q96LA8 1/20 0.47
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
ATM Q13315 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.44
MITF O75030 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
PAX8 Q06710 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CAPN1 P07384 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686299 0.85 ABCG2 (0.67) ABCG2LMNAMAPTATMSMN1; SMN2
SCHEMBL3687299 0.84 ABCG2 (0.47) ABCG2MAPTMEN1KMT2AL3MBTL1
SCHEMBL3684007 0.84 ABCG2 (0.47) ABCG2MAPTMEN1KMT2AL3MBTL1
SCHEMBL4854287 0.78 PTPN1 (0.55) PTPN1ABCG2IDH1ABCB1UGT1A1
SCHEMBL3684939 0.75 TNFRSF1A (0.54) ABCG2LMNAMAPTATMSMN1; SMN2
SCHEMBL3687801 0.74 TNFRSF1A (0.67) ABCG2LMNAMAPTSMN1; SMN2MEN1
SCHEMBL5915314 0.74 PTPN1 (0.50) PTPN1ABCG2IDH1ABCB1UGT1A1
SCHEMBL5915399 0.73 ABCG2 (0.63) PTPN1ABCG2LMNAMAPTATM
SCHEMBL3687310 0.73 ABCG2 (0.67) ABCG2LMNAMAPTATMSMN1; SMN2
SCHEMBL3693509 0.73 ABCG2 (0.67) ABCG2LMNAMAPTATMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed