SCHEMBL3684258

SCHEMBL3684258

COc1ccc(C(=O)C=Cc2cc(N3CCN(C)CC3)ccc2-c2ccccc2C)c(CN(C)C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.45
ABCB1 P08183 2/20 0.40
APP P05067 1/20 0.39
MMP1 P03956 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
ADAM17 P78536 1/20 0.38
HTR6 P50406 1/20 0.37
ABCG2 Q9UNQ0 2/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
F10 P00742 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692597 0.92 TACR1 (0.43) TACR1ABCB1APPMMP1MMP9
SCHEMBL3684257 0.92 TACR1 (0.43) TACR1ABCB1APPMMP1MMP9
SCHEMBL3688891 0.90 TACR1 (0.47) TACR1HTR6CSF1R
SCHEMBL3685079 0.85 ABCB1 (0.43) TACR1ABCB1APPMMP1MMP9
SCHEMBL3685019 0.83 ABCB1 (0.41) TACR1ABCB1APPMMP1MMP9
SCHEMBL3688890 0.83 TACR1 (0.47) TACR1HTR6CSF1R
SCHEMBL3690805 0.83 TACR1 (0.47) TACR1HTR6CSF1R
SCHEMBL3685078 0.81 ALDH1A1 (0.42) TACR1ABCB1MAPTMEN1KMT2A
SCHEMBL3697634 0.81 ALDH1A1 (0.42) TACR1ABCB1MAPTMEN1KMT2A
SCHEMBL3687063 0.80 ALDH1A1 (0.40) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP claimed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed