SCHEMBL3685019

SCHEMBL3685019

COc1ccc(C(=O)C=Cc2cc(-c3ccccc3C)cc(N3CCCN(C)CC3)c2)c(CN(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.41
APP P05067 2/20 0.40
F10 P00742 5/20 0.38
TACR1 P25103 1/20 0.38
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
LMNA P02545 1/20 0.36
RECQL P46063 1/20 0.36
ATM Q13315 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HDAC3 O15379 4/20 0.36
HDAC4 P56524 4/20 0.36
HDAC1 Q13547 4/20 0.36
HDAC7 Q8WUI4 4/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC10 Q969S8 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3685079 0.97 ABCB1 (0.43) ABCB1APPTACR1NPC1MAPT
SCHEMBL3690147 0.91 HDAC3 (0.42) ABCB1TACR1HDAC3HDAC4HDAC1
SCHEMBL3684786 0.87 ABCB1 (0.45) ABCB1APPNPC1MAPTRAB9A
SCHEMBL3687417 0.87 HDAC3 (0.45) ABCB1TACR1HDAC3HDAC4HDAC1
SCHEMBL3687063 0.86 ALDH1A1 (0.40) F10NPC1MAPTRAB9AMEN1
SCHEMBL3685016 0.86 ALDH1A1 (0.40) F10NPC1MAPTRAB9AMEN1
SCHEMBL3684258 0.83 TACR1 (0.45) ABCB1APPF10TACR1MAPT
SCHEMBL3685078 0.83 ALDH1A1 (0.42) ABCB1TACR1NPC1MAPTRAB9A
SCHEMBL3697634 0.83 ALDH1A1 (0.42) ABCB1TACR1NPC1MAPTRAB9A
SCHEMBL3684257 0.80 TACR1 (0.43) ABCB1APPF10TACR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP claimed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed