SCHEMBL3685016

SCHEMBL3685016

COc1ccc(/C=C/C(=O)c2cc(-c3ccccc3C)cc(N3CCCN(C)CC3)c2)c(CN(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
KMT2A Q03164 1/20 0.40
RELA Q04206 1/20 0.40
F10 P00742 9/20 0.39
SMYD2 Q9NRG4 1/20 0.38
KEAP1 Q14145 2/20 0.36
NFE2L2 Q16236 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3687063 1.00 ALDH1A1 (0.40) ALDH1A1MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL3697634 0.97 ALDH1A1 (0.42) ALDH1A1MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL3685078 0.97 ALDH1A1 (0.42) ALDH1A1MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL3690144 0.91 HDAC3 (0.39) ALDH1A1MAPTKDM4EMEN1HPGD
SCHEMBL3692712 0.91 HDAC3 (0.39) ALDH1A1MAPTKDM4EMEN1HPGD
SCHEMBL3684784 0.87 MAPT (0.44) ALDH1A1MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL3689895 0.87 MAPT (0.44) ALDH1A1MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL3697882 0.87 HDAC3 (0.41) ALDH1A1MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL3687415 0.87 HDAC3 (0.41) ALDH1A1MAPTSMN1; SMN2KDM4EMEN1
SCHEMBL3685019 0.86 ABCB1 (0.41) ALDH1A1MAPTMEN1KMT2AF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed