SCHEMBL3685489

SCHEMBL3685489

CC(=O)c1ccccc1NCCCN(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
GLA P06280 1/20 0.49
BRCA1 P38398 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HIF1A Q16665 1/20 0.47
ALDH1A1 P00352 2/20 0.45
PKM P14618 1/20 0.45
BRD4 O60885 1/20 0.44
ATAD2 Q6PL18 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
SLC2A1 P11166 1/20 0.43
APOBEC3A P31941 1/20 0.43
RAD52 P43351 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
CHRNA7 P36544 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686730 0.90 KDM4E (0.47) KDM4EGLAALDH1A1BRD4ATAD2
SCHEMBL10849986 0.84 KMT2A (0.52) KDM4EGLABRCA1SMN1; SMN2HIF1A
Hydrochloric Acid SCHEMBL10847603 0.82 KMT2A (0.51) KDM4EGLABRCA1SMN1; SMN2HIF1A
SCHEMBL6532561 0.81 CNR2 (0.56) KDM4EGLAALDH1A1HPGDHSD17B10
SCHEMBL12767048 0.80 POLB (0.54) SMN1; SMN2ALDH1A1HSD17B10NPC1POLB
SCHEMBL14470975 0.78 KDM4E (0.51) KDM4EGLAALDH1A1HPGDHSD17B10
SCHEMBL1499558 0.78 ALDH1A1 (0.56) KDM4ESMN1; SMN2ALDH1A1HPGDNPC1
SCHEMBL1499550 0.77 TSHR (0.58) KDM4EALDH1A1PKMHPGDHSD17B10
SCHEMBL13033163 0.77 KDM4E (0.51) KDM4EGLASMN1; SMN2ALDH1A1HPGD
SCHEMBL18474174 0.76 SYK (0.53) KDM4EGLAALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed