SCHEMBL3685663

SCHEMBL3685663

CN1CCN(c2ccc(Br)c(C=O)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
GAA P10253 3/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
GLA P06280 1/20 0.47
KDM4E B2RXH2 4/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HTR3A P46098 1/20 0.46
MAPT P10636 3/20 0.45
PTK2B Q14289 2/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
RECQL P46063 1/20 0.45
ADRA2C P18825 2/20 0.44
GFER P55789 1/20 0.43
ESR2 Q92731 1/20 0.43
SIRT6 Q8N6T7 3/20 0.42
HTR1D P28221 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15475184 0.87 ALDH1A1 (0.56) ALDH1A1GAAKMT2AMEN1GLA
SCHEMBL29126321 0.83 GAA (0.52) ALDH1A1GAAKMT2AMEN1KDM4E
SCHEMBL15474866 0.82 ALDH1A1 (0.50) ALDH1A1GAAKMT2AMEN1GLA
SCHEMBL3197069 0.81 MAPT (0.61) ALDH1A1GAAKMT2AMEN1GLA
SCHEMBL15448633 0.77 ALDH1A1 (0.56) ALDH1A1GAAKMT2AMEN1GLA
SCHEMBL11262976 0.77 PIK3CD (0.68) ALDH1A1GAAKMT2AMEN1GLA
Hydrochloric Acid SCHEMBL25231967 0.76 PIK3CD (0.66) ALDH1A1GAAKMT2AMEN1GLA
SCHEMBL3685781 0.76 ADORA2A (0.51) ALDH1A1GAAKMT2AMEN1GLA
SCHEMBL3214435 0.76 SIRT6 (0.66) ALDH1A1MAPTMAPK1SIRT6
SCHEMBL15155902 0.75 ALDH1A1 (0.78) ALDH1A1GAAKMT2AMEN1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed