SCHEMBL368604

SCHEMBL368604

NCc1ccc(F)cc1.O=C(O)c1nc2c(N3CCNCC3=O)cc(N3CCNCC3)cn2c(=O)c1O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
IDO2 Q6ZQW0 1/20 0.34
ALDH1A1 P00352 7/20 0.33
HSD17B10 Q99714 6/20 0.33
HPGD P15428 4/20 0.33
LMNA P02545 3/20 0.33
KDM4E B2RXH2 1/20 0.33
HTR6 P50406 1/20 0.32
USP25 Q9UHP3 3/20 0.32
CYP1A2 P05177 6/20 0.32
CYP3A4 P08684 6/20 0.32
CYP2C9 P11712 6/20 0.32
USP2 O75604 5/20 0.32
CYP2C19 P33261 5/20 0.32
HIF1A Q16665 4/20 0.32
CASP1 P29466 4/20 0.32
CASP7 P55210 4/20 0.32
TP53 P04637 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL368368 0.86 ERCC1 (0.39) HSD17B10LMNAUSP25CYP3A4CYP2C9
SCHEMBL368488 0.82 CYP2C9 (0.41) LMNACYP3A4CYP2C9CYP2C19SMN1; SMN2
SCHEMBL368920 0.81 CYP2C9 (0.41) ALDH1A1LMNACYP3A4CYP2C9CYP2C19
SCHEMBL368726 0.80 PSMD14 (0.40) ALDH1A1HSD17B10HPGDLMNAKDM4E
SCHEMBL368702 0.80 CYP2C9 (0.39) HSD17B10HPGDLMNACYP3A4CYP2C9
SCHEMBL367823 0.74 TTK (0.39) ALDH1A1HSD17B10HPGDLMNAKDM4E
SCHEMBL367927 0.74 CYP2C9 (0.43) HSD17B10LMNACYP3A4CYP2C9CYP2C19
SCHEMBL367904 0.72 KCNH2 (0.37) ALDH1A1HSD17B10HPGDLMNAKDM4E
SCHEMBL10070421 0.71 CALCA (0.49) CYP3A4CYP2C9CYP2C19TP53SMN1; SMN2
SCHEMBL368029 0.70 KCNH2 (0.43) HSD17B10LMNACYP2C9MAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593460-A1 7, 9-NITROGEN RADICAL-4-OXO-4H-PYRIDO[L,2-A]PYRIMIDINE-2-CARBOXYLIC ACID BENZYLAMIDE ANTI-VIRALS Avexa Limited (AU) 2013-05-22 EP disclosed
WO-2012006680-A1 7, 9-NITROGEN RADICAL-4-OXO-4H-PYRIDO[L,2-A]PYRIMIDINE-2-CARBOXYLIC ACID BENZYLAMIDE ANTI-VIRALS AVEXA LIMITED (AU) 2012-01-19 WO disclosed