SCHEMBL3686285

SCHEMBL3686285

CCCN(CC(C)OS(=O)(=O)c1ccc(C)cc1)S(=O)(=O)c1sc2ccc(F)cc2c1C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 7/20 0.36
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PER2 O15055 3/20 0.34
CRY1 Q16526 3/20 0.34
CRY2 Q49AN0 3/20 0.34
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PFKFB4 Q16877 1/20 0.32
GHSR Q92847 1/20 0.31
KAT8 Q9H7Z6 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
SLC2A1 P11166 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692931 0.90 CMA1 (0.35) CMA1LMNAMEN1KMT2APER2
SCHEMBL3686964 0.89 NPSR1 (0.45) CMA1NPSR1L3MBTL1PFKFB4SLC2A1
SCHEMBL3685852 0.85 CMA1 (0.38) CMA1LMNAMEN1KMT2ANPSR1
SCHEMBL13509407 0.85 CMA1 (0.35) CMA1LMNAMEN1KMT2APER2
SCHEMBL6269450 0.83 CMA1 (0.38) CMA1LMNAMEN1KMT2APER2
SCHEMBL13508348 0.81 PER2 (0.43) CMA1LMNAMEN1KMT2APER2
SCHEMBL13508284 0.80 PER2 (0.48) CMA1PER2CRY1CRY2PFKFB4
SCHEMBL3690605 0.79 NPSR1 (0.45) CMA1NPSR1L3MBTL1PFKFB4SLC2A1
SCHEMBL3687739 0.76 SLC2A1 (0.44) CMA1NPSR1L3MBTL1PFKFB4SLC2A1
SCHEMBL3687742 0.76 SLC2A1 (0.44) CMA1NPSR1L3MBTL1PFKFB4SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7655641-B2 Sulfonamide derivatives as PPAR modulators ELI LILLY AND COMPANY (US) 2010-02-02 US disclosed
US-7655641-B2 Sulfonamide derivatives as PPAR modulators ELI LILLY AND COMPANY (US) 2010-02-02 US disclosed
EP-1597248-B1 SULFONAMIDE DERIVATIVES AS PPAR MODULATORS LILLY CO ELI (US) 2007-12-26 EP disclosed
US-20060217433-A1 Sulfonamide derivatives as ppar modulators ELI LILLY AND COMPANY (US) 2006-09-28 US disclosed
EP-1597248-A2 SULFONAMIDE DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-11-23 EP disclosed
WO-2004073606-A2 SULFONAMIDE DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2004-09-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060217433-A1 Sulfonamide derivatives as ppar modulators PPARD, PPARA, PPARG CMA1 4529/4885LMNA 3056/4885MEN1 4858/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.