SCHEMBL3687405

SCHEMBL3687405

Cc1ccccc1-c1ccc(N2CCN(C)CC2)c(/C=C/C(=O)c2cccc(NC(=O)CN(C)C)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
MEN1 O00255 7/20 0.40
KMT2A Q03164 7/20 0.40
LMNA P02545 7/20 0.40
ALDH1A1 P00352 6/20 0.40
MAPT P10636 5/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
RAB9A P51151 4/20 0.40
RECQL P46063 2/20 0.40
NR1H4 Q96RI1 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3687409 1.00 NPC1 (0.41) NPC1MEN1KMT2ALMNAALDH1A1
SCHEMBL3684393 0.91 MAPT (0.45) NPC1MEN1KMT2ALMNAALDH1A1
SCHEMBL3684395 0.91 MAPT (0.45) NPC1MEN1KMT2ALMNAALDH1A1
SCHEMBL3687288 0.85 BCHE (0.42) NPC1MEN1KMT2ALMNAALDH1A1
SCHEMBL3691047 0.80 MEN1 (0.37) NPC1MEN1KMT2ALMNAALDH1A1
SCHEMBL3691987 0.80 LMNA (0.50) MEN1KMT2ALMNAALDH1A1MAPT
SCHEMBL3691989 0.80 LMNA (0.50) MEN1KMT2ALMNAALDH1A1MAPT
SCHEMBL4856323 0.80 LMNA (0.46) NPC1MEN1KMT2ALMNAALDH1A1
SCHEMBL4856336 0.80 LMNA (0.46) NPC1MEN1KMT2ALMNAALDH1A1
SCHEMBL3686504 0.78 HSP90AA1 (0.41) MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed