SCHEMBL3687747

SCHEMBL3687747

NC(=O)c1ccc2[nH]c3c(c2c1)CCCC3C1CCOCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.52
SIRT1 Q96EB6 12/20 0.48
HTR1B P28222 2/20 0.48
SIRT2 Q8IXJ6 5/20 0.47
SIRT3 Q9NTG7 2/20 0.47
RECQL P46063 1/20 0.47
MAPT P10636 2/20 0.45
ALOX15 P16050 2/20 0.45
HTR1A P08908 1/20 0.45
HTR1D P28221 1/20 0.45
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4091350 0.77 BRD3 (0.57) SIRT1SIRT2
SCHEMBL4159842 0.74 DHODH (0.66) MAPKAPK2SIRT1HTR1BSIRT2SIRT3
SCHEMBL5467992 0.73 RB1 (0.62) MAPKAPK2SIRT1HTR1BSIRT2SIRT3
SCHEMBL6447738 0.70 F2 (0.74) MAPKAPK2HTR1BMAPTHTR1AHTR1D
SCHEMBL29643283 0.70 F2 (0.74) MAPKAPK2HTR1BMAPTHTR1AHTR1D
Oxalic Acid SCHEMBL9336199 0.69 BRD3 (0.46) MAPKAPK2SIRT1SIRT2SIRT3RECQL
SCHEMBL5454077 0.69 CDC42 (0.58) MAPKAPK2SIRT1HTR1BSIRT2SIRT3
SCHEMBL5458948 0.69 BRD3 (0.55) MAPKAPK2MAPTALOX15MAPK1SMN1; SMN2
SCHEMBL6238342 0.68 MAPKAPK2 (1.00) MAPKAPK2SIRT1HTR1BHTR1AHTR1D
SCHEMBL30833215 0.68 KCNH2 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190838-A1 CANNABINOID RECEPTOR LIGANDS AstraZeneca AB (SE) 2010-06-02 EP claimed
WO-2009024819-A1 CANNABINOID RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2009-02-26 WO claimed
EP-2190838-A1 CANNABINOID RECEPTOR LIGANDS AstraZeneca AB (SE) 2010-06-02 EP disclosed
WO-2009024819-A1 CANNABINOID RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2009-02-26 WO disclosed