SCHEMBL3687874

SCHEMBL3687874

COc1cccc2c(C(CO)N3CCC[C@H](CNCC=Cc4ccccc4)C3)ccnc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
ENPP1 P22413 1/20 0.32
HTT P42858 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
CTSK P43235 1/20 0.32
PDGFRB P09619 1/20 0.32
PIK3CD O00329 1/20 0.31
PIK3R1 P27986 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
RAB9A P51151 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5652545 0.85 CYP2D6 (0.40) ADRA1AALDH1A1KMT2ATSHROPRM1
SCHEMBL3685798 0.82 HTR1A (0.38) HTR1AADRA1DADRA1AADRA1BENPP1
SCHEMBL5267681 0.71 SLC2A1 (0.47)
SCHEMBL5267677 0.71 SLC2A1 (0.47)
SCHEMBL3697149 0.70 HTR1A (0.35) HTR1AADRA1DADRA1AADRA1BALDH1A1
SCHEMBL13145818 0.69 SLC2A1 (0.49)
SCHEMBL3687873 0.69 SLC2A1 (0.49)
SCHEMBL3688489 0.67 HTR1A (0.33) HTR1AADRA1DADRA1AADRA1BALDH1A1
SCHEMBL3694585 0.65 ADORA2A (0.42) HTR1AADRA1DADRA1AADRA1BENPP1
SCHEMBL3687413 0.65 ADORA2A (0.42) HTR1AADRA1DADRA1AADRA1BENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed
EP-1551829-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2005-07-13 EP disclosed
WO-2004035569-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2004-04-29 WO disclosed