SCHEMBL3690455

SCHEMBL3690455

COC(=O)c1cn2cc(-c3cn[nH]c3)cc(C(F)(F)F)c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.37
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
MAP3K5 Q99683 1/20 0.37
MARK3 P27448 1/20 0.36
HPGD P15428 2/20 0.36
CASP1 P29466 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TSHR P16473 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ROCK2 O75116 4/20 0.36
ROCK1 Q13464 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LCK P06239 1/20 0.35
PTK6 Q13882 1/20 0.35
AURKB Q96GD4 1/20 0.35
CASP7 P55210 1/20 0.35
CLK1 P49759 1/20 0.35
CLK2 P49760 1/20 0.35
KHK P50053 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690539 0.87 RXFP1 (0.38) MAP3K5MARK3ROCK2ROCK1LCK
SCHEMBL3693642 0.79 SCN9A (0.38) MARK3ROCK2ROCK1LCKPTK6
SCHEMBL1583304 0.79 NOTUM (0.41) NOTUMALDH1A1KDM4EHPGDCASP1
SCHEMBL13261951 0.79 AURKB (0.35) MAP3K5MARK3ROCK2ROCK1LCK
Hydrochloric Acid SCHEMBL3695164 0.79 SCN9A (0.37) MARK3ROCK2ROCK1LCKPTK6
SCHEMBL3687179 0.78 SCN9A (0.42) ROCK2ROCK1LCKPTK6AURKB
SCHEMBL3684324 0.78 AURKB (0.36) ALDH1A1KDM4EMARK3HPGDCASP1
SCHEMBL1583390 0.77 RXFP1 (0.47) NOTUMALDH1A1KDM4ESMN1; SMN2MAPT
SCHEMBL1583985 0.77 NOTUM (0.40) NOTUMALDH1A1KDM4EHPGDCASP1
SCHEMBL1583885 0.77 ROCK2 (0.39) NOTUMALDH1A1KDM4EHPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections GLAXOSMITHKLINE LLC 2012-05-17 US disclosed
EP-2187883-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2010-05-26 EP disclosed
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections GLAXOSMITHKLINE LLC 2009-07-09 US disclosed
WO-2009023179-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2009-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections OAT, HAVCR2, CPS1 NOTUM 1173/4885ALDH1A1 1337/4885KDM4E 2131/4885
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections OAT, HAVCR2, CPS1 NOTUM 1173/4885ALDH1A1 1337/4885KDM4E 2131/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.