SCHEMBL3690891

SCHEMBL3690891

CN1C(=O)Cc2ccc(-c3ccc(C[C@H](NC(=O)C4CCCCN4C(=O)O)C(N)=O)cc3)cc21

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
VHL P40337 1/20 0.52
CTSC P53634 8/20 0.48
CTSK P43235 2/20 0.48
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
XIAP P98170 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7858105 0.89 VHL (0.47) VHLCTSCCTSKOPRM1OPRD1
SCHEMBL3701201 0.86 CTSC (0.65) CTSCCTSK
SCHEMBL2075246 0.80 VHL (0.51) VHLOPRM1OPRD1OPRK1XIAP
SCHEMBL2073451 0.80 VHL (0.51) VHLCTSCOPRM1OPRD1OPRK1
SCHEMBL3692633 0.78 VHL (0.57) VHLOPRM1OPRD1OPRK1XIAP
SCHEMBL4398641 0.77 VHL (0.51) VHLOPRM1OPRD1OPRK1XIAP
SCHEMBL2071996 0.77 VHL (0.54) VHLOPRM1OPRD1OPRK1XIAP
SCHEMBL2072259 0.76 VHL (0.48) VHLOPRM1OPRD1OPRK1XIAP
SCHEMBL7857586 0.76 CTSC (0.60) CTSCCTSK
SCHEMBL2074016 0.76 CTSC (0.51) VHLCTSCOPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010142985-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL]PIPERIDIN-2-YLCARBOXMIDE COMPOUNDS 761 ASTRAZENECA AB (SE) 2010-12-16 WO disclosed