SCHEMBL3695006

SCHEMBL3695006

COc1ccccc1-c1ccc(C(=O)/C=C/c2ccccc2CN(C)C)c(N2CCCN(C)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.44
DRD2 P14416 3/20 0.41
DRD3 P35462 3/20 0.41
DRD4 P21917 2/20 0.41
HRH2 P25021 2/20 0.41
HRH1 P35367 1/20 0.41
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
HIF1A Q16665 1/20 0.39
KEAP1 Q14145 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3693463 1.00 PTPN1 (0.44) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3685244 0.97 PTPN1 (0.43) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3686258 0.97 PTPN1 (0.43) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3691194 0.91 PTPN1 (0.41) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3693464 0.91 PTPN1 (0.43) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3684550 0.91 PTPN1 (0.41) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3686127 0.90 PTPN1 (0.41) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3685873 0.90 PTPN1 (0.41) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3685247 0.87 ALDH1A1 (0.43) PTPN1DRD2DRD3DRD4HRH2
SCHEMBL3681834 0.87 HDAC3 (0.46) PTPN1ALDH1A1LMNASMN1; SMN2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed